SCHEMBL7420115

SCHEMBL7420115

CCCc1c(C=O)c2ccc(C(=O)NS(=O)(=O)c3ccccc3)cc2n1Cc1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
FLT1 P17948 2/20 0.40
FLT4 P35916 2/20 0.40
KDR P35968 2/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
TP53 P04637 1/20 0.39
PPARG P37231 1/20 0.39
GNRHR P30968 1/20 0.39
CCR2 P41597 1/20 0.39
AGTR2 P50052 1/20 0.39
EGLN3 Q9H6Z9 1/20 0.39
PTGES O14684 1/20 0.38
ROCK2 O75116 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7418847 0.88 L3MBTL1 (0.41) FLT1FLT4KDRTP53PPARG
SCHEMBL7421444 0.87 KMT2A (0.54) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL7418980 0.84 MAPT (0.47) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL7462431 0.84 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL7417407 0.80 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL7420372 0.79 KMT2A (0.56) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL7421704 0.79 PPARG (0.38) FLT1FLT4KDRPPARGCCR2
SCHEMBL7473116 0.77 MAPT (0.48) ALDH1A1MEN1KMT2ALMNAGAA
SCHEMBL5882017 0.77 CCR2 (0.48) FLT1FLT4KDRGAATP53
SCHEMBL7418878 0.77 ALDH1A1 (0.53) ALDH1A1MEN1KMT2ALMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820441-B1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO (JP) 2002-06-26 EP disclosed
US-6358992-B1 Method of inhibiting neoplastic cells with indole derivatives CELL PATHWAYS, INC. 2002-03-19 US disclosed
US-6069156-A Indole derivatives as cGMP-PDE inhibitors FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-05-30 US disclosed
EP-0820441-A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-01-28 EP disclosed
WO-1996032379-A1 INDOLE DERIVATIVES AS cGMP-PDE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-10-17 WO disclosed