SCHEMBL7420191

SCHEMBL7420191

CC(C)(C[CH]C(=O)N(Cc1ccccc1)C1(C#N)CCNC1)C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SNCA P37840 2/20 0.34
CTSS P25774 4/20 0.32
CTSK P43235 2/20 0.32
CTSB P07858 3/20 0.31
OPRM1 P35372 2/20 0.31
CTSL P07711 2/20 0.31
RIPK1 Q13546 2/20 0.31
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416904 0.94 SNCA (0.35) SNCACTSSCTSKCTSBOPRM1
SCHEMBL7021618 0.83 SNCA (0.34) SNCACTSSCTSKCTSLCYP2D6
SCHEMBL7017468 0.82
SCHEMBL7020795 0.81
SCHEMBL7417847 0.80 OPRM1 (0.38) OPRM1
SCHEMBL7420196 0.78 CTSS (0.36) SNCACTSSCTSKCTSBOPRM1
SCHEMBL7417804 0.78 CTSS (0.32) CTSSCTSKOPRM1
SCHEMBL7425513 0.78 CTSS (0.31) CTSS
SCHEMBL7415538 0.78 ADRA1D (0.32) SNCACTSSCTSKCYP2D6SLC6A2
SCHEMBL7018594 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed