SCHEMBL7420439

SCHEMBL7420439

O=C(OCc1ccc(OCc2ccccc2)cc1)C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.58
NR4A1 P22736 1/20 0.57
NR4A2 P43354 1/20 0.57
NR4A3 Q92570 1/20 0.57
FFAR1 O14842 1/20 0.56
FFAR4 Q5NUL3 1/20 0.56
PTGS1 P23219 2/20 0.54
PTGS2 P35354 2/20 0.54
LMNA P02545 1/20 0.54
CYP1A2 P05177 1/20 0.54
SLC6A2 P23975 1/20 0.54
CYP2C19 P33261 1/20 0.54
SLC6A3 Q01959 1/20 0.54
HIF1A Q16665 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
PARP10 Q53GL7 1/20 0.54
LTA4H P09960 1/20 0.53
LAP3 P28838 1/20 0.53
SRD5A2 P31213 1/20 0.53
ALOX5 P09917 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3296385 0.88 ALDH1A1 (0.57) LMNASLC6A2SLC6A3ALDH1A1L3MBTL1
SCHEMBL27923357 0.87 ALDH1A1 (0.55) LMNASLC6A2SLC6A3ALDH1A1L3MBTL1
SCHEMBL13686681 0.84 PRKCA (0.66) MAOBNR4A1NR4A2NR4A3FFAR1
Acetic Acid SCHEMBL27401419 0.83 ALDH1A1 (0.61) MAOBLMNASLC6A2SLC6A3ALDH1A1
SCHEMBL9258815 0.83 CA1 (0.47) MAOBSLC6A2SLC6A3HDAC6ALDH1A1
Trimethylammonium SCHEMBL27550267 0.82 ALDH1A1 (0.55) LMNASLC6A2CYP2C19SLC6A3ALDH1A1
Dimethylamine SCHEMBL27585618 0.82 KMT2A (0.55) LMNASLC6A2SLC6A3ALDH1A1SMN1; SMN2
SCHEMBL8333346 0.82 NR4A1 (0.66) MAOBNR4A1NR4A2NR4A3FFAR1
Trifluoroacetic Acid SCHEMBL7420441 0.81 FFAR1 (0.60) MAOBNR4A1NR4A2NR4A3FFAR1
SCHEMBL2381708 0.81 CES1 (0.69) MAOBNR4A1NR4A2NR4A3FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021411-A1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LIMITED (GB) 2000-07-26 EP disclosed
WO-1997022589-A1 BENZAMIDE DERIVATIVES AS THROMBIN INHIBITORS GLAXO GROUP LIMITED (GB) 1997-06-26 WO disclosed