SCHEMBL7420754

SCHEMBL7420754

CCOC(=O)CC(=O)CC(O)c1ccc(OC)c(OC2CCCC2)c1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 12/20 0.52
PDE4B Q07343 11/20 0.52
PDE4D Q08499 10/20 0.52
PDE4C Q08493 9/20 0.52
STAT3 P40763 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7928933 0.87 PDE4A (0.57) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL6889943 0.87 PDE4A (0.60) PDE4APDE4BPDE4DPDE4C
SCHEMBL7175088 0.81 PDE4A (0.65) PDE4APDE4BPDE4DPDE4C
SCHEMBL7320061 0.78 PDE4A (0.48) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL8770917 0.77 ACHE (0.48) PDE4APDE4BPDE4DPDE4CSTAT3
SCHEMBL9283831 0.77 PDE4B (0.53) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7357352 0.76 PDE4B (0.53) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL7913418 0.76 PDE4A (0.59) PDE4APDE4BPDE4DPDE4C
SCHEMBL6229209 0.76 PDE4B (0.50) PDE4APDE4BPDE4DPDE4CPOLB
SCHEMBL2988958 0.76 PDE4A (0.63) PDE4APDE4BPDE4DPDE4CPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248769-B1 ANTIINFLAMMATORY AGENT EURO-CELTIQUE S.A. (LU) 2001-06-19 US disclosed
US-6103749-A PHENYL IMIDAZOLE COMPOUNDS USEFUL FOR TREATMENT OF ASTHMA, ALLERGIES, INFLAMMATION AND DEPRESSION EURO-CELTIQUE S.A. (LU) 2000-08-15 US disclosed
US-5922751-A BRONCHODILATOR AND ANTIINFLAMMATORY AGENT WITHOUT UNDESIRABLE CARDIOVASCULAR STIMULATION CAUSED BY PHOSPHODIESTERASE III INHIBITOR EURO-CELTIQUE, S.A. (LU) 1999-07-13 US disclosed
EP-0766676-A4 COMPOUNDS FOR AND METHOD OF INHIBITING PHOSPHODIESTERASE IV EURO CELTIQUE SA (LU) 1998-07-08 EP disclosed
EP-0766676-A1 COMPOUNDS FOR AND METHOD OF INHIBITING PHOSPHODIESTERASE IV Euroceltique S.A. (LU) 1997-04-09 EP disclosed
WO-1996000218-A1 COMPOUNDS FOR AND METHOD OF INHIBITING PHOSPHODIESTERASE IV EURO-CELTIQUE, S.A. (LU) 1996-01-04 WO disclosed