SCHEMBL7420977

SCHEMBL7420977

CC(NCc1ccc(Br)cc1)[Si](C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 1/20 0.43
CTSK P43235 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
AGER Q15109 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13858736 0.82 SIGMAR1 (0.59) SIGMAR1MEN1KMT2AMAPTTAAR1
SCHEMBL2548456 0.79 PYCR1 (0.48) PYCR1CTSKSIGMAR1NPC1RAB9A
SCHEMBL11693602 0.74 SIGMAR1 (0.46) PYCR1CTSKSIGMAR1NPC1RAB9A
SCHEMBL3833687 0.73 SIGMAR1 (0.79) SIGMAR1CYP1A2CYP2D6LMNATAAR1
SCHEMBL5854794 0.73 IDO1 (0.38) PYCR1CTSKNPC1RAB9ACYP1A2
SCHEMBL17605856 0.70 PYCR1 (0.44) PYCR1CTSKSIGMAR1NPC1RAB9A
SCHEMBL13041050 0.70 SMN1; SMN2 (0.70) CYP1A2CYP2D6CYP2C19MEN1KMT2A
SCHEMBL21966166 0.70 PYCR1 (0.41) PYCR1CTSKSIGMAR1NPC1RAB9A
SCHEMBL9288254 0.70 AGER (0.61) NPC1RAB9AMEN1KMT2AL3MBTL1
SCHEMBL17605180 0.70 PYCR1 (0.44) PYCR1CTSKSIGMAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934265-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF Du Pont Pharmaceuticals Company (US) 1999-08-11 EP disclosed
WO-1998006694-A1 AMIDINOPHENYL-PYRROLIDINES, -PYRROLINES, AND -ISOXAZOLIDINES AND DERIVATIVES THEREOF DU PONT PHARMACEUTICALS COMPANY (US) 1998-02-19 WO disclosed