SCHEMBL7422329

SCHEMBL7422329

COC(=O)[C@H](Cc1ccc(-c2c(C)cc[nH]c2=O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.48
ITGB7 P26010 2/20 0.48
KLK5 Q9Y337 1/20 0.46
CTSS P25774 6/20 0.46
CTSK P43235 5/20 0.46
EPHX2 P34913 1/20 0.42
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
ACE P12821 1/20 0.40
BCL2 P10415 1/20 0.40
TACR1 P25103 1/20 0.40
AKT1 P31749 1/20 0.39
SCN9A Q15858 1/20 0.39
PTPN1 P18031 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535596 0.85 ITGA4 (0.48) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7421167 0.83 ITGA4 (0.46) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7415719 0.83 ITGA4 (0.46) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL6235727 0.81 ITGA4 (0.54) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL1822923 0.80 CTSS (0.58) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL10033679 0.79 CTSS (0.69) KLK5CTSSCTSKCTSLCTSB
SCHEMBL1826757 0.79 CTSS (0.69) KLK5CTSSCTSKCTSLCTSB
SCHEMBL2802961 0.79 CTSS (0.69) KLK5CTSSCTSKCTSLCTSB
SCHEMBL13651745 0.79 KLK5 (0.58) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL12035376 0.79 KLK5 (0.58) ITGA4ITGB7KLK5CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed