SCHEMBL7415719

SCHEMBL7415719

COC(=O)[C@H](Cc1ccc(-c2c(C)c(Cl)c[nH]c2=O)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.46
ITGB7 P26010 2/20 0.46
KLK5 Q9Y337 1/20 0.44
CTSS P25774 6/20 0.44
CTSK P43235 5/20 0.44
TACR1 P25103 2/20 0.40
EPHX2 P34913 1/20 0.40
CTSL P07711 2/20 0.39
CTSB P07858 1/20 0.39
SCN9A Q15858 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
BCL2 P10415 3/20 0.38
ACE P12821 1/20 0.38
AKT1 P31749 1/20 0.38
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7421167 0.89 ITGA4 (0.46) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7420188 0.86 KLK5 (0.49) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7535596 0.85 ITGA4 (0.48) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7422329 0.83 ITGA4 (0.48) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL7417736 0.80 ITGB1 (0.54) ITGA4ITGB7
SCHEMBL7416021 0.79 GPR142 (0.40) ITGA4ITGB7
Hydrochloric Acid SCHEMBL7420715 0.79 ALDH1A1 (0.39) ITGA4ITGB7AKT1
SCHEMBL7411842 0.78 ITGB1 (0.55) ITGA4ITGB7
SCHEMBL14885702 0.78 CTSS (0.54) ITGA4ITGB7KLK5CTSSCTSK
SCHEMBL14885705 0.78 CTSS (0.54) ITGA4ITGB7KLK5CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244625-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2002-10-02 EP disclosed
WO-2001042215-A1 4-PYRIDINYL-N-ACYL-L-PHENYLALANINES F. HOFFMANN-LA ROCHE AG (CH) 2001-06-14 WO disclosed