SCHEMBL7423519

SCHEMBL7423519

N=C(N)NCC(CN)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 2/20 0.49
GABBR1 Q9UBS5 2/20 0.49
BCAT2 O15382 1/20 0.42
TAAR1 Q96RJ0 4/20 0.42
HTR2A P28223 2/20 0.42
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
AOC3 Q16853 3/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KDM4E B2RXH2 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7518330 0.84 BCAT2 (0.41) GABBR2GABBR1BCAT2TAAR1HTR2A
Hydrochloric Acid SCHEMBL6947022 0.80 GABBR2 (0.56) GABBR2GABBR1BCAT2MTNR1AMTNR1B
SCHEMBL20773797 0.80 GABBR2 (0.59) GABBR2GABBR1BCAT2TAAR1HTR2A
SCHEMBL3921879 0.78 BCAT2 (0.68) BCAT2TAAR1CYP2D6SMN1; SMN2AOC3
SCHEMBL21408380 0.78 GBA1 (0.46) BCAT2AOC3KDM4EL3MBTL1
SCHEMBL14769096 0.78 BCAT2 (0.68) BCAT2TAAR1CYP2D6SMN1; SMN2AOC3
SCHEMBL1985542 0.77 MTNR1A (0.69) GABBR2GABBR1BCAT2TAAR1HTR2A
SCHEMBL4018230 0.76 AOC3 (0.58) BCAT2TAAR1SMN1; SMN2AOC3
SCHEMBL17198959 0.76 AOC3 (0.58) BCAT2TAAR1SMN1; SMN2AOC3
SCHEMBL1983010 0.76 NPC1 (0.63) GABBR2GABBR1BCAT2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4709032-A VASODILATION AND HYPOTENSIVE AGENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-11-24 US disclosed
US-4634770-A VASODILATORS, HYPOTENSIVES ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1987-01-06 US disclosed
EP-0109023-A1 Isoquinolinesulfonamide derivatives and process for the preparation thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-05-23 EP disclosed