SCHEMBL7424464

SCHEMBL7424464

COc1cc(CC(=O)Nc2ccc(C(CC(=O)O)N(C)S(=O)(=O)c3cccnc3)nc2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.56
ITGA4 P13612 10/20 0.56
HPGD P15428 3/20 0.41
ALDH1A1 P00352 1/20 0.41
AHR P35869 1/20 0.40
RAB9A P51151 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7590998 0.89 ITGB1 (0.62) ITGB1ITGA4MEN1KMT2APOLB
SCHEMBL7379255 0.89 ITGA4 (0.45) ITGB1ITGA4AHRRAB9AKMT2A
SCHEMBL7379944 0.87 ITGB1 (0.54) ITGB1ITGA4HPGDALDH1A1MEN1
SCHEMBL7422070 0.87 ITGB1 (0.59) ITGB1ITGA4AHRMEN1KMT2A
SCHEMBL7379263 0.86 ITGA4 (0.55) ITGB1ITGA4MEN1KMT2A
SCHEMBL7426753 0.85 ITGB1 (0.64) ITGB1ITGA4MEN1KMT2APOLB
SCHEMBL7422320 0.85 ITGA4 (0.56) ITGB1ITGA4MEN1KMT2A
SCHEMBL7647170 0.83 ITGA4 (0.62) ITGB1ITGA4MEN1KMT2A
SCHEMBL7417458 0.83 ITGA4 (0.49) ITGB1ITGA4HPGDALDH1A1AHR
SCHEMBL7421722 0.83 ITGB1 (0.61) ITGB1ITGA4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479519-B1 INHIBITORS OF CELL ADHESION; TREATMENT OF ASTHMA OR INFLAMMATORY BOWEL DISEASE AVENTIS PHARMA LIMITED (GB) 2002-11-12 US disclosed
EP-1027328-A1 SUBSTITUTED ANILIDES Aventis Pharma Limited (GB) 2000-08-16 EP disclosed
WO-1999023063-A1 SUBSTITUTED ANILIDES AVENTIS PHARMA LIMITED (GB) 1999-05-14 WO disclosed