SCHEMBL7424674

SCHEMBL7424674

N#Cc1cccc(CN2CC[C@H](NC(=O)c3ccccc3)C2=O)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
BRD4 O60885 1/20 0.48
SRC P12931 3/20 0.48
FAAH O00519 1/20 0.47
FNTA P49354 5/20 0.46
FNTB P49356 5/20 0.46
PGGT1B P53609 5/20 0.46
KCNH2 Q12809 2/20 0.46
F10 P00742 4/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
CCR3 P51677 1/20 0.45
CYP3A4 P08684 1/20 0.45
NPY1R P25929 1/20 0.44
NTRK1 P04629 1/20 0.44
ACKR3 P25106 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417098 0.91 ROCK2 (0.47) HDAC1HDAC8HDAC6BRD4SRC
SCHEMBL7420184 0.91 SRC (0.49) HDAC1HDAC8HDAC6BRD4SRC
SCHEMBL7421293 0.91 BRD4 (0.47) HDAC1HDAC8HDAC6BRD4SRC
SCHEMBL7428971 0.90 BRD4 (0.48) HDAC1HDAC8HDAC6BRD4FNTA
SCHEMBL7423020 0.90 CCR3 (0.46) HDAC1HDAC8HDAC6BRD4FNTA
SCHEMBL7422293 0.89 BRD4 (0.50) HDAC1HDAC8HDAC6BRD4SRC
SCHEMBL7418733 0.89 CCKBR (0.52) HDAC1HDAC8HDAC6BRD4F10
SCHEMBL7418566 0.88 F10 (0.47) BRD4FNTAFNTBPGGT1BKCNH2
SCHEMBL7419869 0.88 MCHR1 (0.49) BRD4SRCF10CCR3
SCHEMBL7418602 0.88 SRC (0.48) HDAC1HDAC8HDAC6BRD4SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853618-A4 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE POULENC RORER PHARMA (US) 2000-03-15 EP disclosed
EP-0853618-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N- (AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1998-07-22 EP disclosed
WO-1996040679-A1 SUBSTITUTED (SULFINIC ACID, SULFONIC ACID, SULFONYLAMINO OR SULFINYLAMINO) N-[(AMINOIMINOMETHYL)PHENYLALKYL]-AZAHETEROCYCLYLAMIDE COMPOUNDS RHÔNE-POULENC RORER PHARMACEUTICALS INC. (US) 1996-12-19 WO disclosed