SCHEMBL7425433

SCHEMBL7425433

COc1cc(N(CCC2CCN(CCC(=O)O)CC2)C(C)=O)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.52
ITGB1 P05556 5/20 0.45
ITGA4 P13612 5/20 0.45
THRB P10828 1/20 0.42
OPRM1 P35372 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
CCR3 P51677 1/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426905 0.95 ACHE (0.51) ACHEITGB1ITGA4OPRM1
SCHEMBL7430185 0.93 ITGB1 (0.45) ACHEITGB1ITGA4THRBSIGMAR1
SCHEMBL7431414 0.92 ACHE (0.54) ACHEITGB1ITGA4SIGMAR1MEN1
SCHEMBL7539587 0.91 ACHE (0.47) ACHEITGB1ITGA4OPRM1SIGMAR1
SCHEMBL7393503 0.87 ACHE (0.49) ACHEITGB1ITGA4SIGMAR1CCR3
SCHEMBL7428874 0.86 ACHE (0.47) ACHEITGB1ITGA4MEN1GAA
SCHEMBL7424847 0.86 ITGB1 (0.46) ITGB1ITGA4THRBOPRM1SIGMAR1
SCHEMBL7425014 0.84 ACHE (0.46) ACHEITGB1ITGA4CCR3MEN1
SCHEMBL7425039 0.84 ITGB1 (0.54) ACHEITGB1ITGA4SIGMAR1MEN1
SCHEMBL7422232 0.84 THRB (0.46) ITGB1ITGA4THRBSIGMAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed