SCHEMBL7425604

SCHEMBL7425604

Clc1nc(Cl)c2cc(-n3cccn3)ccc2n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.50
NLRP3 Q96P20 3/20 0.41
HRH3 Q9Y5N1 1/20 0.40
RORC P51449 6/20 0.40
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAT2A P31153 1/20 0.39
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
ADORA2A P29274 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778095 0.75 NOTUM (0.56) NOTUMNLRP3MAPK1KDM4EALDH1A1
SCHEMBL3974447 0.73 HRH3 (0.53) NOTUMNLRP3HRH3MAPK1KDM4E
SCHEMBL1536322 0.72 NOTUM (0.51) NOTUMNLRP3HRH3MAPK1KDM4E
SCHEMBL11337325 0.71 NOTUM (0.63) NOTUMMAPK1KDM4EALDH1A1DRD2
SCHEMBL12450338 0.71 NOTUM (0.53) NOTUMNLRP3MAPK1KDM4EALDH1A1
SCHEMBL23667579 0.70 KDM4E (0.57) NOTUMNLRP3HRH3MAPK1KDM4E
SCHEMBL3760506 0.70 TERT (0.50) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL28740983 0.70 NOTUM (0.49) NOTUMNLRP3HRH3MAPK1KDM4E
SCHEMBL12575851 0.70 NLRP3 (0.43) NOTUMNLRP3HRH3RORCLMNA
SCHEMBL28046310 0.69 NCOA3 (0.56) NOTUMNLRP3HRH3MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691967-B1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO LTD (JP) 1998-09-02 EP disclosed
US-5707998-A CYCLIC-GMP PHOSPHODIESTERASE INHIBITORS, TREATING CARDIOVASCULAR DISORDERS AND ASTHMA EISAI CO., LTD. (JP) 1998-01-13 US disclosed
EP-0691967-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS Eisai Co., Ltd. (JP) 1996-01-17 EP disclosed
WO-1994022855-A1 NITROGEN-CONTAINING FUSED-HETEROCYCLE COMPOUNDS EISAI CO., LTD. (JP) 1994-10-13 WO disclosed