SCHEMBL7425720

SCHEMBL7425720

CCOC(=O)c1ccc2c(cnn2C(C=O)N(C)OC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 4/20 0.39
SIRT1 Q96EB6 3/20 0.39
NPC1 O15118 3/20 0.38
MAPT P10636 2/20 0.38
NLRP3 Q96P20 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
RAB9A P51151 5/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HSD17B2 P37059 1/20 0.37
THRB P10828 1/20 0.37
ALDH1A1 P00352 3/20 0.36
PPARG P37231 1/20 0.36
NCOA2 Q15596 1/20 0.36
NCOA1 Q15788 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4123693 0.80 EZH2 (0.51) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL7425711 0.74 POLB (0.42) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL3436319 0.73 CCNC (0.49) SIRT2SIRT1NPC1MAPTCA12
SCHEMBL8682160 0.73 HSD17B10 (0.40) SIRT2SIRT1NPC1MAPTCA12
Hydrochloric Acid SCHEMBL8683788 0.73 ALDH1A1 (0.40) SIRT2SIRT1NPC1MAPTNLRP3
Hydrochloric Acid SCHEMBL8683796 0.73 ALDH1A1 (0.40) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL904672 0.72 MAPT (0.48) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL4959328 0.72 MAOA (0.43) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL7426706 0.71 CHEK1 (0.56) SIRT2SIRT1NPC1MAPTNLRP3
SCHEMBL7426302 0.70 EGFR (0.45) NPC1MAPTNLRP3CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054871-A2 PYRIMIDINES AND TRIAZINES AS INTEGRIN ANTAGONISTS Du Pont Pharmaceuticals Company (US) 2000-11-29 EP disclosed
WO-1999050249-A2 PYRIMIDINES AND TRIAZINES AS INTEGRIN ANTAGONISTS DU PONT PHARMACEUTICALS COMPANY (US) 1999-10-07 WO disclosed