SCHEMBL7426619

SCHEMBL7426619

CC(C)(C)OC(=O)N[C@](C)(C(=O)NO)c1ccco1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
MAPT P10636 3/20 0.41
HTT P42858 2/20 0.41
KMT2A Q03164 5/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288246 0.70 NPC1 (0.41) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL7769259 0.70 KMT2A (0.42) NPC1RAB9ASMN1; SMN2MAPTKMT2A
SCHEMBL16279155 0.69 MAPT (0.49) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL16279156 0.69 MAPT (0.49) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL5124451 0.68 SMN1; SMN2 (0.52) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL28793821 0.67 RAB9A (0.62) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL12666543 0.66 MEN1 (0.41) NPC1RAB9AMAPTKMT2AALDH1A1
SCHEMBL14152450 0.66 TDP1 (0.36) NPC1RAB9ASMN1; SMN2KMT2AMEN1
SCHEMBL28968872 0.65 MAPT (0.42) NPC1RAB9ASMN1; SMN2MAPTHTT
SCHEMBL2953752 0.65 CA12 (0.47) NPC1RAB9AKMT2ACTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6018020-A VIRICIDES WHICH ARE PROTEASE INHIBITORS AGAINST HEPATITIS C AND HEPATITIS G HOFFMAN-LA ROCHE INC. (US) 2000-01-25 US disclosed
EP-0941233-A2 ANTIVIRAL PEPTIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-09-15 EP disclosed
US-5866684-A Peptidyl inhibitors of viral proteases HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1998022496-A2 ANTIVIRAL PEPTIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1998-05-28 WO disclosed