SCHEMBL7427630

SCHEMBL7427630

Fc1ccc(C(c2ccc(F)cc2)N2CCCNCC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.59
CYP19A1 P11511 1/20 0.59
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
ACHE P22303 3/20 0.53
OPRD1 P41143 8/20 0.50
OPRM1 P35372 2/20 0.49
OPRK1 P41145 2/20 0.49
P4HB P07237 2/20 0.47
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
SLC6A3 Q01959 2/20 0.46
SIGMAR1 Q99720 1/20 0.44
OPRL1 P41146 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336219 0.93 CYP2D6 (0.67) CYP2D6CYP19A1MEN1KMT2AACHE
SCHEMBL16225886 0.86 MEN1 (0.79) CYP2D6CYP19A1MEN1KMT2AOPRD1
SCHEMBL1138318 0.86 MEN1 (0.79) CYP2D6CYP19A1MEN1KMT2AOPRD1
SCHEMBL1138320 0.86 MEN1 (0.79) CYP2D6CYP19A1MEN1KMT2AOPRD1
SCHEMBL8182035 0.85 CYP2D6 (0.57) CYP2D6CYP19A1MEN1KMT2AACHE
SCHEMBL11193886 0.83 CYP2D6 (0.56) CYP2D6CYP19A1MEN1KMT2AACHE
SCHEMBL8479321 0.82 MEN1 (0.85) CYP2D6CYP19A1MEN1KMT2AOPRD1
Acetic Acid SCHEMBL27992925 0.82 OPRD1 (0.65) CYP2D6CYP19A1MEN1KMT2AOPRD1
SCHEMBL16226147 0.82 MEN1 (0.67) CYP2D6CYP19A1MEN1KMT2AOPRD1
SCHEMBL14280201 0.81 ACHE (0.71) MEN1KMT2AACHEOPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661148-A ANTIHYPOXIC AGENT FOR RESPIRATORY SYSTEM DISORDER TEIJIN LIMITED (JP) 1997-08-26 US disclosed
EP-0514540-B1 PYRROLO 2,3-d]PYRIMIDINE DERIVATIVE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL PREPARATION COMPRISING THE DERIVATIVE AS ACTIVE INGREDIENT TEIJIN LTD (JP) 1996-07-17 EP disclosed
EP-0283310-B1 N-BENZHYDRYL-SUBSTITUTED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-05-26 EP disclosed
EP-0514540-A1 PYRROLO 2,3-d]PYRIMIDINE DERIVATIVE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL PREPARATION COMPRISING THE DERIVATIVE AS ACTIVE INGREDIENT TEIJIN LIMITED (JP) 1992-11-25 EP disclosed
US-5028610-A Calcium Channel Blockers SANKYO COMPANY LIMITED (JP) 1991-07-02 US disclosed
EP-0283310-A1 N-Benzhydryl-substituted heterocyclic derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-09-21 EP disclosed