SCHEMBL7428115

SCHEMBL7428115

CC(=O)C(Br)C(=O)c1ccncc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
TP53 P04637 1/20 0.44
LMNA P02545 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
PTGS2 P35354 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
MPO P05164 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CYP2A6 P11509 1/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL330589 0.79 L3MBTL1 (0.48) NAPRTCYP3A4LMNAALDH1A1MEN1
SCHEMBL1887807 0.79 CYP1A2 (0.51) NAPRTCYP1A2CYP3A4TP53LMNA
SCHEMBL5353045 0.79 GSK3B (0.56) NAPRTCYP1A2CYP3A4LMNAALDH1A1
SCHEMBL7432886 0.78 NAPRT (0.46) NAPRTCYP1A2CYP3A4TP53LMNA
Bromide SCHEMBL4188500 0.78 CYP1A2 (0.50) NAPRTCYP1A2CYP3A4TP53LMNA
SCHEMBL15458715 0.78 ALDH1A1 (0.48) LMNAALDH1A1MEN1KMT2AHPGD
SCHEMBL1881302 0.77 KMT2A (0.45) CYP1A2CYP3A4LMNAALDH1A1MEN1
SCHEMBL908908 0.76 CES2 (0.46) ALDH1A1MEN1KMT2AHPGDHTT
SCHEMBL19104772 0.76 CYP1A2 (0.49) NAPRTCYP1A2CYP3A4TP53LMNA
SCHEMBL7933884 0.75 NAPRT (0.48) NAPRTCYP1A2CYP3A4TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0329070-B1 Cardiotonic alkanoyl and aroyl oxazolones MERRELL DOW PHARMA (US) 1994-01-05 EP disclosed
US-4866182-A TREATMENT OF HEART FAILURE MERRELL DOW PHARMACEUTICALS INC. (US) 1989-09-12 US disclosed
EP-0329070-A1 Cardiotonic alkanoyl and aroyl oxazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1989-08-23 EP disclosed