SCHEMBL7428797

SCHEMBL7428797

O=C(O)NC(CC(=O)NC1CCCNC[C@@H]1O)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPN1 P15169 2/20 0.38
CPB2 Q96IY4 2/20 0.38
ALDH1A1 P00352 4/20 0.33
SLC6A1 P30531 2/20 0.33
SLC6A11 P48066 1/20 0.33
TSHR P16473 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC6A13 Q9NSD5 1/20 0.33
KMT2A Q03164 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM3 P20309 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
EPHX1 P07099 1/20 0.31
CYP2C19 P33261 2/20 0.31
CYP2C9 P11712 1/20 0.31
MAPT P10636 1/20 0.31
CYP3A4 P08684 1/20 0.30
HPGD P15428 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591617 0.84 HDAC4 (0.38) CPN1CPB2EPHX1
SCHEMBL4769116 0.74 CPB2 (0.42) CPN1CPB2CYP3A4
SCHEMBL4769110 0.74 CPB2 (0.42) CPN1CPB2CYP3A4
SCHEMBL4769131 0.74 CPN1 (0.40) CPN1CPB2SLC6A1SLC6A11TSHR
SCHEMBL7428804 0.74 CPN1 (0.40) CPN1CPB2SLC6A1SLC6A11TSHR
SCHEMBL3956518 0.73 CYP2C9 (0.33) CPN1CPB2ALDH1A1SLC6A1SLC6A11
SCHEMBL7421894 0.73 CPN1 (0.32) CPN1CPB2ALDH1A1SLC6A1SLC6A11
SCHEMBL6592080 0.72 PSEN1 (0.37) CPN1CPB2ALDH1A1SLC6A1SLC6A11
SCHEMBL22233331 0.71 CPN1 (0.50) CPN1CPB2SLC6A1SLC6A11TSHR
SCHEMBL3956504 0.70 CTSK (0.40) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed