SCHEMBL7429046

SCHEMBL7429046

COc1ccc(-c2cc(OC)ccc2C(=O)Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.58
KDM4E B2RXH2 1/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
BACE1 P56817 3/20 0.50
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
CYP3A4 P08684 1/20 0.46
MAPK1 P28482 1/20 0.46
PRKAB2 O43741 1/20 0.45
PRKAG1 P54619 1/20 0.45
PRKAA2 P54646 1/20 0.45
PRKAA1 Q13131 1/20 0.45
PRKAG3 Q9UGI9 1/20 0.45
PRKAG2 Q9UGJ0 1/20 0.45
PRKAB1 Q9Y478 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7591657 0.84 SMN1; SMN2 (0.75) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL4131227 0.83 GAA (0.57) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL7502103 0.81 NPC1 (0.66) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL11197823 0.80 NPC1 (0.55) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL5631648 0.79 MAPT (0.55) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL7083789 0.77 SMN1; SMN2 (0.64) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL4392160 0.77 NPC1 (0.53) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL8566031 0.77 SMN1; SMN2 (0.64) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL9151080 0.77 SMN1; SMN2 (0.64) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9
SCHEMBL9683222 0.77 SMN1; SMN2 (0.64) SMN1; SMN2KDM4ECYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183239-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2002-03-06 EP disclosed
WO-2000069821-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed