SCHEMBL7429230

SCHEMBL7429230

COc1cc(CC(=O)N2CCCC2c2cc(CCC(=O)O)on2)ccc1OCc1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.45
NPC1 O15118 8/20 0.45
KMT2A Q03164 3/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
MEN1 O00255 1/20 0.40
APP P05067 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432425 0.94 MEN1 (0.47) RAB9ANPC1KMT2AMEN1APP
SCHEMBL27570769 0.93 APP (0.43) RAB9ANPC1KMT2AMEN1APP
SCHEMBL27570763 0.93 FFAR1 (0.44) RAB9ANPC1KMT2AMEN1APP
SCHEMBL7583778 0.92 FFAR1 (0.44) RAB9ANPC1KMT2AMEN1APP
SCHEMBL7481227 0.90 RAB9A (0.41) RAB9ANPC1KMT2AMEN1LMNA
SCHEMBL27570770 0.90 S1PR1 (0.47) RAB9ANPC1
SCHEMBL27570759 0.88 GRM5 (0.43) RAB9ANPC1KMT2AMEN1APP
SCHEMBL7439258 0.88 S1PR1 (0.41) RAB9ANPC1APPSMN1; SMN2HPGD
SCHEMBL7435979 0.87 CPT1A (0.43) RAB9ANPC1SMN1; SMN2HPGD
SCHEMBL7429711 0.87 FFAR4 (0.42) KMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1413210-A Non-peptidyl inhibitors of VLA-4 dependent cell binding for the treatment of inflammation, autoimmune diseases and respiratory diseases PFIZER PROD INC (US) 2003-04-23 CN disclosed
EP-1244656-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2002-10-02 EP disclosed
WO-2001051487-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2001-07-19 WO disclosed