SCHEMBL7439258

SCHEMBL7439258

CCOc1cc(CC(=O)N2CCCC2c2cc(CCC(=O)O)on2)ccc1OCc1ccc(OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
APP P05067 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CHRM1 P11229 4/20 0.38
SCD O00767 2/20 0.38
SCD5 Q86SK9 1/20 0.38
FFAR1 O14842 1/20 0.38
CPT1A P50416 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27570769 0.95 APP (0.43) APPNPC1RAB9ASCDSCD5
SCHEMBL7432425 0.89 MEN1 (0.47) APPNPC1RAB9A
SCHEMBL7429230 0.88 RAB9A (0.45) SMN1; SMN2APPNPC1RAB9AHPGD
SCHEMBL7583778 0.88 FFAR1 (0.44) SMN1; SMN2APPNPC1RAB9AFFAR1
SCHEMBL27570759 0.84 GRM5 (0.43) APPNPC1RAB9AFFAR1ALDH1A1
SCHEMBL27570763 0.84 FFAR1 (0.44) APPNPC1RAB9AFFAR1
SCHEMBL27578899 0.83 NPC1 (0.44) NPC1RAB9ASCDSCD5FFAR1
SCHEMBL7422672 0.83 FFAR1 (0.48) NPC1RAB9AFFAR1ALDH1A1
SCHEMBL7433078 0.83 FFAR1 (0.42) NPC1RAB9AFFAR1CPT1A
SCHEMBL7487553 0.83 FFAR1 (0.42) NPC1RAB9AFFAR1CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244656-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2002-10-02 EP disclosed
WO-2001051487-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2001-07-19 WO disclosed