SCHEMBL7429752

SCHEMBL7429752

CN1C2CCCC1CC(NC(=O)c1c(O)c3ccccc3n(-c3ccccc3)c1=O)C2

nearest known ligand 0.96

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 9/20 0.96
HTR3E A5X5Y0 5/20 0.96
HTR3B O95264 5/20 0.96
HTR3D Q70Z44 5/20 0.96
HTR3C Q8WXA8 5/20 0.96
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
GAA P10253 1/20 0.59
PPARG P37231 1/20 0.59
NCOA2 Q15596 1/20 0.59
SLC22A2 O15244 1/20 0.57
CHRNB2 P17787 1/20 0.57
CHRNA3 P32297 1/20 0.57
CHRNA4 P43681 1/20 0.57
KCNH2 Q12809 1/20 0.57
SLC47A1 Q96FL8 1/20 0.57
ALDH1A1 P00352 1/20 0.51
CYP3A4 P08684 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430349 0.98 HTR3A (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7436991 0.83 HTR3A (0.74) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7439804 0.79 HTR3E (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7430595 0.78 HTR3A (0.67) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9556624 0.78 HTR3A (0.64) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9556621 0.78 HTR3A (0.64) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9556956 0.78 HTR3A (0.64) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7435767 0.78 HTR3A (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7444121 0.77 NPC1 (0.71) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL9556583 0.74 HTR3A (0.62) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed