SCHEMBL7444121

SCHEMBL7444121

CN1C2CCCC1CC(NC(=O)c1c(O)c3ccccc3[nH]c1=O)C2

nearest known ligand 0.94

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.71
MEN1 O00255 3/20 0.71
KMT2A Q03164 3/20 0.71
RAB9A P51151 3/20 0.70
SMN1; SMN2 Q16637 2/20 0.70
POLB P06746 1/20 0.70
RXFP1 Q9HBX9 1/20 0.70
HTR3E A5X5Y0 5/20 0.66
HTR3B O95264 5/20 0.66
HTR3A P46098 5/20 0.66
HTR3D Q70Z44 5/20 0.66
HTR3C Q8WXA8 5/20 0.66
KDM4E B2RXH2 4/20 0.59
NLRP3 Q96P20 1/20 0.59
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
SLC22A2 O15244 1/20 0.53
CHRNB2 P17787 1/20 0.53
CHRNA3 P32297 1/20 0.53
CHRNA4 P43681 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435902 0.97 KMT2A (0.72) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL1622809 0.83 RAB9A (1.00) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL22639784 0.83 RAB9A (1.00) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7308018 0.81 HTR3A (0.50) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7300915 0.78 HTR3E (0.52) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7430312 0.78 HTR3A (0.58) MEN1KMT2ASMN1; SMN2HTR3EHTR3B
SCHEMBL13597998 0.78 KMT2A (0.82) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7301719 0.77 HTR3E (0.51) NPC1MEN1KMT2ARAB9ASMN1; SMN2
SCHEMBL7429752 0.77 HTR3A (0.96) NPC1RAB9AHTR3EHTR3BHTR3A
SCHEMBL10673661 0.76 HTR3A (0.78) RAB9ASMN1; SMN2HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed