SCHEMBL7429758

SCHEMBL7429758

Nc1ccc2c3c(cccc13)C(=O)N(C1CCN(Cc3ccccc3)CC1)C2=O

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.57
USP2 O75604 3/20 0.50
KMT2A Q03164 3/20 0.50
KEAP1 Q14145 3/20 0.50
NFE2L2 Q16236 3/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
HTT P42858 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
OPRM1 P35372 1/20 0.47
OPRK1 P41145 1/20 0.47
OPRL1 P41146 1/20 0.47
MEN1 O00255 2/20 0.47
ATM Q13315 2/20 0.47
CYP1B1 Q16678 2/20 0.47
CHRM3 P20309 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13016528 0.87 ACHE (0.67) ACHESMN1; SMN2OPRM1OPRK1OPRL1
Hydrochloric Acid SCHEMBL9585539 0.84 ACHE (0.50) ACHEOPRM1OPRK1OPRL1CHRM3
SCHEMBL9586632 0.83 ACHE (0.64) ACHEKMT2AKDM4EALDH1A1MAPT
SCHEMBL250673 0.83 ACHE (0.69) ACHEOPRM1OPRK1OPRL1CHRM3
Hydrochloric Acid SCHEMBL9585516 0.82 ACHE (0.63) ACHEKMT2AKDM4EALDH1A1MAPT
SCHEMBL9585353 0.81 USP2 (0.61) USP2KMT2AKEAP1NFE2L2KDM4E
SCHEMBL7646060 0.79 KEAP1 (0.57) USP2KMT2AKEAP1NFE2L2KDM4E
SCHEMBL9586240 0.77 USP2 (0.58) USP2KMT2AKEAP1NFE2L2KDM4E
SCHEMBL8327851 0.75 ACHE (0.57) ACHEKMT2ACHRM3
SCHEMBL9585526 0.75 HTR1A (0.49) ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5202318-A Antiserotonine, antiemetic agents SYNTEX (U.S.A.) INC. (US) 1993-04-13 US disclosed
WO-1992021673-A1 NOVEL AZABICYCLOBENZISOQUINOLINES SYNTEX (U.S.A.) INC. (US) 1992-12-10 WO disclosed