SCHEMBL7430261

SCHEMBL7430261

COC(=O)c1ccc(N2CCCC2)c(NC(=O)C(CSC(C)=O)Cc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.52
ALDH1A1 P00352 5/20 0.52
MAPT P10636 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
HPGD P15428 2/20 0.47
MEN1 O00255 2/20 0.47
GAA P10253 1/20 0.46
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ABCC3 O15438 1/20 0.45
NR1I2 O75469 1/20 0.45
ABCB11 O95342 1/20 0.45
NR3C1 P04150 1/20 0.45
RARG P13631 1/20 0.45
CNR1 P21554 1/20 0.45
OPRK1 P41145 1/20 0.45
NR1H2 P55055 1/20 0.45
PPARA Q07869 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435482 0.92 KMT2A (0.56) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL7438991 0.92 MAPT (0.49) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL7432434 0.91 MAPT (0.48) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL7431823 0.79 KDM4E (0.49) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL7427411 0.77 CYP2D6 (0.43) KMT2AALDH1A1CYP1A2CYP3A4MEN1
SCHEMBL7440859 0.77 ALDH1A1 (0.51) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL7433764 0.76 KMT2A (0.50) KMT2AALDH1A1MAPTHPGDMEN1
SCHEMBL7433938 0.76 PPARA (0.50) KMT2AALDH1A1CYP1A2CYP3A4MEN1
SCHEMBL7435502 0.76 CYP1A2 (0.58) KMT2AALDH1A1MAPTCYP1A2CYP3A4
SCHEMBL10779210 0.75 CYP1A2 (0.49) ALDH1A1CYP1A2CYP3A4HPGDCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed