SCHEMBL7435482

SCHEMBL7435482

COC(=O)c1ccc(N2CCOCC2)c(NC(=O)C(CSC(C)=O)Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.56
ALDH1A1 P00352 9/20 0.52
HPGD P15428 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
HSD17B10 Q99714 1/20 0.52
POLB P06746 1/20 0.50
CYP1A2 P05177 2/20 0.47
CYP3A4 P08684 2/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 1/20 0.47
KDM4E B2RXH2 1/20 0.46
TSHR P16473 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GAA P10253 2/20 0.44
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
ABCC3 O15438 1/20 0.43
NR1I2 O75469 1/20 0.43
ABCB11 O95342 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430261 0.92 KMT2A (0.52) KMT2AALDH1A1HPGDSMN1; SMN2CYP1A2
SCHEMBL7438991 0.84 MAPT (0.49) KMT2AALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL7432434 0.83 MAPT (0.48) KMT2AALDH1A1HPGDHSD17B10POLB
SCHEMBL7432199 0.78 ALDH1A1 (0.56) KMT2AALDH1A1HPGDSMN1; SMN2HSD17B10
SCHEMBL7370831 0.74 CYP1A2 (0.52) KMT2AALDH1A1SMN1; SMN2CYP1A2CYP3A4
SCHEMBL7433938 0.74 PPARA (0.50) KMT2AALDH1A1POLBCYP1A2CYP3A4
SCHEMBL7435502 0.73 CYP1A2 (0.58) KMT2AALDH1A1HPGDSMN1; SMN2CYP1A2
SCHEMBL10779210 0.73 CYP1A2 (0.49) ALDH1A1HPGDSMN1; SMN2CYP1A2CYP3A4
SCHEMBL7442246 0.72 CYP1A2 (0.50) KMT2AALDH1A1CYP1A2CYP3A4MEN1
SCHEMBL7425603 0.72 CYP1A2 (0.50) KMT2AALDH1A1POLBCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed