SCHEMBL7431016

SCHEMBL7431016

COc1cccc(-c2c(OC)cccc2C(=O)Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.47
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HSD17B1 P14061 1/20 0.46
GPR35 Q9HC97 1/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
HDAC4 P56524 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
FABP3 P05413 1/20 0.44
FABP4 P15090 1/20 0.44
FABP5 Q01469 1/20 0.44
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
DHODH Q02127 1/20 0.42
CNR1 P21554 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796258 0.87 GPR35 (0.55) ERN1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL7430974 0.84 FABP4 (0.58) NPC1TP53RAB9AGAAFABP3
SCHEMBL7894667 0.79 GAA (0.57) KDM4EGAAHDAC4HDAC8POLB
SCHEMBL27940845 0.75 PARP1 (0.58) NPC1TP53RAB9ASMN1; SMN2GPR35
SCHEMBL15782121 0.74 KDM4E (0.53) NPC1RAB9ASMN1; SMN2HSD17B1GPR35
SCHEMBL14585873 0.74 ITGB1 (0.47) TP53RAB9ASMN1; SMN2FABP3FABP4
SCHEMBL9357148 0.74 JAK2 (0.56) NPC1TP53RAB9ASMN1; SMN2KDM4E
SCHEMBL7333428 0.73 ERN1 (0.44) ERN1SMN1; SMN2GAAHDAC4HDAC8
SCHEMBL16712927 0.73 HSD17B2 (0.60) NPC1RAB9AHDAC4HDAC8POLB
Benzene SCHEMBL28272579 0.73 JAK2 (0.55) NPC1TP53RAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183239-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2002-03-06 EP disclosed
WO-2000069821-A1 AROMATIC SULFONE HYDROXAMIC ACID METALLOPROTEASE INHIBITOR G.D. SEARLE & CO. (US) 2000-11-23 WO disclosed