SCHEMBL7433133

SCHEMBL7433133

COc1cc(C(O)CO)ccc1OCCCN1CCC(C(c2ccc(F)cc2F)c2ccc(F)cc2F)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 4/20 0.42
HTR2C P28335 4/20 0.42
HRH1 P35367 4/20 0.42
HTR2B P41595 4/20 0.42
DRD2 P14416 4/20 0.42
DRD4 P21917 3/20 0.42
SLC6A4 P31645 3/20 0.42
HTR6 P50406 3/20 0.42
HTR2A P28223 3/20 0.42
ADRA2C P18825 2/20 0.42
ADRA1A P35348 2/20 0.42
HTR1A P08908 2/20 0.42
ADRA2B P18089 2/20 0.42
KCNH2 Q12809 2/20 0.42
ABCB11 O95342 1/20 0.42
CHRM2 P08172 1/20 0.42
ADRA2A P08913 1/20 0.42
CHRM1 P11229 1/20 0.42
ACHE P22303 1/20 0.42
SLC6A2 P23975 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435553 0.88 ABCB11 (0.45) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7448170 0.87 DRD1 (0.41) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7433432 0.86 DRD2 (0.47) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7436648 0.85 KCNH2 (0.48) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7436929 0.83 ABCB11 (0.51) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7439642 0.82 ABCB11 (0.51) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7448352 0.82 ABCB11 (0.51) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL10558073 0.81 DRD1 (0.45) DRD1HTR2CHRH1HTR2BDRD2
Oxalic Acid SCHEMBL10461422 0.81 ABCB11 (0.58) DRD1HTR2CHRH1HTR2BDRD2
SCHEMBL7432094 0.80 ABCB11 (0.49) DRD1HTR2CHRH1HTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed