SCHEMBL7436648

SCHEMBL7436648

COc1cc(CCO)ccc1OCCCN1CCC(C(c2ccc(F)cc2F)c2ccc(F)cc2F)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.48
TMEM97 Q5BJF2 3/20 0.48
SIGMAR1 Q99720 3/20 0.48
DRD2 P14416 6/20 0.46
HTR2A P28223 5/20 0.46
HTR1A P08908 4/20 0.46
HRH3 Q9Y5N1 3/20 0.46
DRD1 P21728 4/20 0.45
HTR2C P28335 4/20 0.45
HRH1 P35367 4/20 0.45
HTR2B P41595 4/20 0.45
ADRA1B P35368 3/20 0.45
DRD4 P21917 3/20 0.45
SLC6A4 P31645 3/20 0.45
HTR6 P50406 3/20 0.45
HRH2 P25021 2/20 0.45
HTR1D P28221 2/20 0.45
HTR1B P28222 2/20 0.45
HTR7 P34969 2/20 0.45
ADRA1A P35348 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433432 0.93 DRD2 (0.47) KCNH2TMEM97SIGMAR1DRD2HTR2A
SCHEMBL7433713 0.85 HTR1A (0.43) KCNH2SIGMAR1DRD2HTR2AHTR1A
SCHEMBL7443763 0.85 KCNH2 (0.44) KCNH2TMEM97SIGMAR1DRD2HTR2A
SCHEMBL7433133 0.85 DRD1 (0.42) KCNH2TMEM97SIGMAR1DRD2HTR2A
SCHEMBL7436929 0.84 ABCB11 (0.51) KCNH2SIGMAR1DRD2HTR2AHTR1A
SCHEMBL7439642 0.83 ABCB11 (0.51) KCNH2SIGMAR1DRD2HTR2AHTR1A
SCHEMBL7448352 0.82 ABCB11 (0.51) KCNH2SIGMAR1DRD2HTR2AHTR1A
Oxalic Acid SCHEMBL10461422 0.82 ABCB11 (0.58) KCNH2SIGMAR1DRD2HTR2AHTR1A
SCHEMBL7435553 0.82 ABCB11 (0.45) KCNH2SIGMAR1DRD2HTR2AHTR1A
SCHEMBL7432094 0.80 ABCB11 (0.49) KCNH2SIGMAR1DRD2HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed