SCHEMBL7433325

SCHEMBL7433325

O=C(CN1CCN(C(c2ccc(F)cc2)c2ccc(F)cc2)CC1)Nc1cccc2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.63
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
CA7 P43166 3/20 0.56
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 2/20 0.55
GAA P10253 3/20 0.52
MAPT P10636 2/20 0.52
ALPL P05186 1/20 0.52
ALPG P10696 1/20 0.52
CA9 Q16790 1/20 0.52
KMT2A Q03164 6/20 0.51
MEN1 O00255 5/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HSD17B10 Q99714 2/20 0.50
USP2 O75604 1/20 0.50
HPGD P15428 1/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 2/20 0.48
CHRNB2 P17787 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430239 0.79 CA1 (0.65) CYP2C19CA1CA2CA7ALDH1A1
Hydrochloric Acid SCHEMBL7432666 0.78 CA1 (0.64) CYP2C19CA1CA2CA7ALDH1A1
SCHEMBL3833776 0.77 CYP2C19 (0.60) CYP2C19ALDH1A1KDM4EGAAMAPT
SCHEMBL3393276 0.76 SLC27A1 (0.74) CA1CA2CA7ALDH1A1KDM4E
SCHEMBL30585259 0.76 ALDH1A1 (0.73) CYP2C19ALDH1A1KDM4EGAAMAPT
SCHEMBL29078430 0.76 ALDH1A1 (0.73) CYP2C19ALDH1A1KDM4EGAAMAPT
SCHEMBL3395419 0.75 CA1 (0.52) CA1CA2CA7ALDH1A1KDM4E
SCHEMBL23086156 0.75 MEN1 (0.60) CA1CA2CA7ALDH1A1KDM4E
SCHEMBL7423903 0.73 ALOX15 (0.60) CA1CA2CA7ALDH1A1GAA
SCHEMBL31611860 0.73 CYP2C19 (0.73) CYP2C19ALDH1A1KDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283310-B1 N-BENZHYDRYL-SUBSTITUTED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-05-26 EP disclosed
US-5028610-A Calcium Channel Blockers SANKYO COMPANY LIMITED (JP) 1991-07-02 US disclosed
EP-0283310-A1 N-Benzhydryl-substituted heterocyclic derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-09-21 EP disclosed