SCHEMBL7434243

SCHEMBL7434243

CC(C)C[C@H](NC(=O)[C@H](C)N(C(=O)C1CCCC1)c1ccccc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MME P08473 3/20 0.47
ALDH1A1 P00352 1/20 0.45
PSMB5 P28074 3/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.42
CTSL P07711 2/20 0.41
CTSB P07858 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MMP2 P08253 1/20 0.41
MMP7 P09237 1/20 0.41
MMP9 P14780 1/20 0.41
MMP12 P39900 1/20 0.41
MMP13 P45452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693745 0.83 MME (0.53) MMEALDH1A1GAACTSLCTSB
SCHEMBL9831516 0.82 MME (0.50) MMECTSLCTSBCTSSCTSK
SCHEMBL6854264 0.82 MME (0.54) MMECTSLCTSBCTSSCTSK
SCHEMBL27675065 0.79 MME (0.47) MMEALDH1A1CTSLCTSBCTSS
SCHEMBL9829010 0.78 CTSL (0.51) MMECTSLCTSBCTSSCTSK
SCHEMBL10443778 0.78 MME (0.42) MMEALDH1A1GAACTSK
SCHEMBL10443960 0.78 ALDH1A1 (0.42) MMEALDH1A1GAACTSLCTSB
SCHEMBL7275108 0.77 MME (0.47) MMEALDH1A1MAPK1
SCHEMBL21288033 0.77 HTT (0.42) ALDH1A1PSMB5SMN1; SMN2
SCHEMBL1524821 0.76 CTSK (0.52) MMECTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296581-A2 Amino acid 1,2-diketo derivatives as renin inhibitors E.R. SQUIBB & SONS, INC. (US) 1988-12-28 EP disclosed