SCHEMBL7434370

SCHEMBL7434370

CC(C)CCN(C(=O)NCC#N)C(=O)c1cccc(N(CCN2CCOCC2)C(=O)N2CCNCC2)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASR P41180 10/20 0.46
CTSL P07711 4/20 0.36
CTSB P07858 4/20 0.36
CTSS P25774 4/20 0.36
CTSK P43235 4/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MLYCD O95822 1/20 0.34
EPHX2 P34913 2/20 0.34
MC4R P32245 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6186860 0.80 NPC1 (0.47) CASREPHX2
SCHEMBL6182151 0.74 NAMPT (0.44) CTSSMLYCDMC4R
SCHEMBL7482944 0.72 JAK2 (0.43) CTSLCTSBCTSSCTSK
SCHEMBL7482953 0.71 CTSL (0.34) CTSLCTSBCTSSCTSK
SCHEMBL6186854 0.68 NPC1 (0.48) CASREPHX2
Trifluoroacetic Acid SCHEMBL7045149 0.66 CTSL (0.42) CTSLCTSBCTSSCTSKEPHX2
Trifluoroacetic Acid SCHEMBL6183907 0.64 FAAH (0.46)
SCHEMBL6182109 0.64 CTSS (0.46) CTSLCTSBCTSSCTSK
SCHEMBL6183132 0.62 GAA (0.48)
SCHEMBL6182144 0.62 NAMPT (0.46) MLYCDMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed