SCHEMBL7434779

SCHEMBL7434779

CN(C)Cc1nnc2n1-c1ccc(Cl)cc1C(c1ccccn1)=NC2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 4/20 0.74
HPGD P15428 4/20 0.56
GABRA1 P14867 5/20 0.56
GABRA5 P31644 5/20 0.56
GABRA3 P34903 5/20 0.56
GABRA2 P47869 5/20 0.56
GABRB2 P47870 4/20 0.56
LMNA P02545 2/20 0.52
BRD4 O60885 2/20 0.52
CNR1 P21554 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
RECQL P46063 1/20 0.52
PDE4D Q08499 2/20 0.51
GABRG2 P18507 1/20 0.51
HTR2A P28223 1/20 0.51
GABRB3 P28472 1/20 0.51
ADRA1A P35348 1/20 0.51
CYP1A2 P05177 1/20 0.51
KDM4E B2RXH2 1/20 0.49
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11711028 0.92 OPRK1 (0.63) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11830458 0.91 OPRK1 (0.62) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11838524 0.90 OPRK1 (0.61) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11796054 0.90 OPRK1 (0.61) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11830564 0.90 OPRK1 (0.59) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL7425412 0.88 GABRA1 (0.73) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL7440925 0.88 OPRK1 (0.57) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11838526 0.88 OPRK1 (0.57) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11605914 0.88 GABRA1 (0.58) OPRK1HPGDGABRA1GABRA5GABRA3
SCHEMBL11606037 0.88 OPRK1 (0.58) OPRK1HPGDGABRA1GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4001262-A Process for the production of 1-[(dimethylamino)methyl]-6-phenyl-4H-triazolo[4,3-a][1,4]-benzodiazepine THE UPJOHN COMPANY (US) 1977-01-04 US disclosed
US-3995043-A BENZODIAZEPINE DERIVATIVES FOR TREATING ANXIETY AND DEPRESSION THE UPJOHN COMPANY (US) 1976-11-30 US disclosed