SCHEMBL7434824

SCHEMBL7434824

Brc1[c]c2ccc(Br)cc2c(Br)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.33
HSP90AA1 P07900 1/20 0.32
TLR9 Q9NR96 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HTT P42858 1/20 0.32
JAK2 O60674 2/20 0.31
CHEK1 O14757 1/20 0.31
AURKA O14965 1/20 0.31
DAPK3 O43293 1/20 0.31
PRKD3 O94806 1/20 0.31
MAP4K4 O95819 1/20 0.31
PAK4 O96013 1/20 0.31
ABL1 P00519 1/20 0.31
NTRK1 P04629 1/20 0.31
CSF1R P07333 1/20 0.31
RET P07949 1/20 0.31
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7430263 0.76 MEN1 (0.32) ALDH1A1HTT
SCHEMBL7794514 0.70 ALOX15 (0.33) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL1451102 0.67 ESR2 (0.39) ALOX15HSP90AA1ALDH1A1HTT
SCHEMBL598418 0.66 ALOX15 (0.42) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL16158369 0.61 CYP2A6 (0.47) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL7609339 0.61 AHR (0.33) HTTJAK2CHEK1AURKADAPK3
SCHEMBL20356136 0.61 HSP90AA1 (0.46) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL20356135 0.61 ALOX15 (0.37) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL8556469 0.61 CYP2A6 (0.48) ALOX15HSP90AA1TLR9ALDH1A1MAPK1
SCHEMBL1569370 0.59 CYP2A6 (0.52) ALOX15ALDH1A1HTTJAK2CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0283310-B1 N-BENZHYDRYL-SUBSTITUTED HETEROCYCLIC DERIVATIVES, THEIR PREPARATION AND THEIR USE Sankyo Company Limited (JP) 1993-05-26 EP disclosed
US-5028610-A Calcium Channel Blockers SANKYO COMPANY LIMITED (JP) 1991-07-02 US disclosed
EP-0283310-A1 N-Benzhydryl-substituted heterocyclic derivatives, their preparation and their use Sankyo Company Limited (JP) 1988-09-21 EP disclosed