SCHEMBL7435001

SCHEMBL7435001

COc1cc(C(O)C(=O)O)ccc1OCCCN1CCC(C(O)(c2cccc(F)c2)c2cccc(F)c2)CC1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.50
MEN1 O00255 7/20 0.47
KMT2A Q03164 3/20 0.45
LMNA P02545 2/20 0.45
HRH1 P35367 2/20 0.45
DRD3 P35462 2/20 0.45
KCNH2 Q12809 2/20 0.45
CNR1 P21554 1/20 0.45
APEX1 P27695 1/20 0.45
PDE4A P27815 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2B P41595 1/20 0.45
BLM P54132 1/20 0.45
PDE3A Q14432 1/20 0.45
DRD2 P14416 1/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP2J2 P51589 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432529 0.91 PAX8 (0.52) PAX8MEN1KMT2ALMNAHRH1
Water SCHEMBL7428725 0.90 PAX8 (0.51) PAX8MEN1KMT2ALMNAHRH1
SCHEMBL7442321 0.85 PAX8 (0.51) PAX8MEN1KMT2AHRH1DRD3
SCHEMBL10460775 0.85 ABCB11 (0.57) PAX8MEN1KMT2AHRH1DRD3
SCHEMBL7446953 0.84 HRH1 (0.54) PAX8MEN1HRH1DRD3KCNH2
SCHEMBL7446850 0.83 PAX8 (0.51) PAX8MEN1HRH1DRD3KCNH2
SCHEMBL7440209 0.83 MEN1 (0.50) PAX8MEN1KMT2AHRH1KCNH2
Oxalic Acid SCHEMBL7438851 0.82 PAX8 (0.51) PAX8MEN1KMT2ALMNAHRH1
SCHEMBL7438853 0.81 MEN1 (0.49) PAX8MEN1KMT2AHRH1HTR2A
SCHEMBL7443328 0.81 CACNA1B (0.42) PAX8HRH1DRD3KCNH2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed