SCHEMBL9565317

SCHEMBL9565317

CC(C)Cc1nc(-c2cccnc2)n[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
CYP2A6 P11509 3/20 0.42
BTK Q06187 1/20 0.41
ALK Q9UM73 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
METAP2 P50579 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
DYRK1A Q13627 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565348 0.83 SMN1; SMN2 (0.50) SMN1; SMN2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL7435148 0.77 PDGFRB (0.49) CYP2A6ALKKDM5BMETAP2SIRT3
SCHEMBL9565355 0.73 ALDH1A1 (0.49) SMN1; SMN2CYP2A6DYRK1AALDH1A1CYP1A2
SCHEMBL9464649 0.72 NR1H2 (0.47) SMN1; SMN2PRMT5WDR77KDM5BCYP1A2
SCHEMBL1435798 0.70 SMN1; SMN2 (0.63) SMN1; SMN2PRKAA1CYP2A6BTKALK
SCHEMBL9565323 0.70 HSD17B10 (0.45) SMN1; SMN2CYP2A6ALDH1A1CYP1A2CYP3A4
SCHEMBL11598851 0.69 SMN1; SMN2 (0.87) SMN1; SMN2CYP2A6BTKALDH1A1CYP1A2
SCHEMBL7440831 0.68 CYP2A6 (0.44) CYP2A6ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL831106 0.67 SMN1; SMN2 (0.63) SMN1; SMN2CYP2A6BTKMETAP2SIRT3
SCHEMBL4873033 0.67 SMN1; SMN2 (0.63) SMN1; SMN2CYP2A6BTKALKMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543245-A1 Renin inhibiting amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1993-05-26 EP disclosed