SCHEMBL7435235

SCHEMBL7435235

COc1ccc(CCCC(=O)N[C@@](O)(C(=O)O)[C@H](N)C(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.54
KMT2A Q03164 1/20 0.54
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAB9A P51151 1/20 0.46
ALOX5 P09917 1/20 0.45
POLB P06746 1/20 0.44
PLAAT3 P53816 1/20 0.44
PLAAT5 Q96KN8 1/20 0.44
PLAAT2 Q9NWW9 1/20 0.44
PLAAT4 Q9UL19 1/20 0.44
F2RL1 P55085 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431314 0.87 HPGD (0.41) ALDH1A1KMT2AHPGD
SCHEMBL10509298 0.87 TRPV1 (0.46) ALDH1A1KMT2AHPGDPLAAT3PLAAT5
SCHEMBL5057819 0.87 HPGD (0.52) ALDH1A1HPGDRAB9AALOX5POLB
SCHEMBL5807162 0.87 HPGD (0.52) ALDH1A1HPGDRAB9AALOX5POLB
SCHEMBL851962 0.82 ALDH1A1 (0.43) ALDH1A1KMT2AHPGDRAB9A
SCHEMBL7432238 0.80 ALDH1A1 (0.54) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL11412947 0.79 HDAC2 (0.46) ALDH1A1KMT2AHPGDRAB9A
SCHEMBL7436219 0.78 ALDH1A1 (0.55) ALDH1A1KMT2ARAB9AALOX5POLB
SCHEMBL13902990 0.73 ALDH1A1 (0.63) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL11405396 0.73 HDAC1 (0.53) HPGDRAB9AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed