SCHEMBL7436219

SCHEMBL7436219

COc1ccc(CCCC(=O)N[C@@](O)(C(=O)O)[C@H](NC(=O)OCc2ccccc2)C(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
KMT2A Q03164 1/20 0.55
ATM Q13315 1/20 0.48
CTSL P07711 2/20 0.47
CTSS P25774 2/20 0.47
CTSK P43235 2/20 0.47
CASP1 P29466 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
PLAAT3 P53816 1/20 0.44
PLAAT5 Q96KN8 1/20 0.44
PLAAT2 Q9NWW9 1/20 0.44
PLAAT4 Q9UL19 1/20 0.44
CAPN1 P07384 1/20 0.44
CAPN2 P17655 1/20 0.44
RAB9A P51151 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ACHE P22303 1/20 0.43
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438359 0.93 CASP1 (0.49) ALDH1A1KMT2AATMCTSLCTSS
SCHEMBL7435235 0.78 ALDH1A1 (0.54) ALDH1A1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL25465074 0.73 CTRB1 (0.57) ATMCTSLCTSSCTSK
SCHEMBL12442117 0.73 CTRB1 (0.57) ATMCTSLCTSSCTSK
SCHEMBL29337555 0.72 ALDH1A1 (0.53) ALDH1A1KMT2AATMCTSLCTSS
SCHEMBL5057819 0.72 HPGD (0.52) ALDH1A1HDAC8RAB9APOLBALOX5
SCHEMBL5807162 0.72 HPGD (0.52) ALDH1A1HDAC8RAB9APOLBALOX5
SCHEMBL8569421 0.72 ALDH1A1 (0.65) ALDH1A1KMT2AATMCTSLCTSS
SCHEMBL2406036 0.72 ALDH1A1 (0.65) ALDH1A1KMT2AATMCTSLCTSS
SCHEMBL15506190 0.72 ALDH1A1 (1.00) ALDH1A1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed