SCHEMBL7435247

SCHEMBL7435247

CSc1ccc(C(=O)O)cc1N

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 12/20 0.57
ALDH1A1 P00352 8/20 0.57
TDP1 Q9NUW8 4/20 0.57
AR P10275 1/20 0.51
MAPT P10636 9/20 0.49
GAA P10253 8/20 0.49
HPGD P15428 6/20 0.49
THRB P10828 3/20 0.49
GFER P55789 2/20 0.49
HTT P42858 1/20 0.49
PLEC Q15149 1/20 0.49
CDC25B P30305 1/20 0.46
HSD17B10 Q99714 5/20 0.45
L3MBTL1 Q9Y468 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
GLA P06280 1/20 0.45
RCE1 Q9Y256 1/20 0.45
POLB P06746 2/20 0.44
LMNA P02545 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275002 0.85 CDC25B (0.50) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL858819 0.85 AR (0.54) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL6517360 0.84 KDM4E (0.60) KDM4EALDH1A1TDP1MAPTGAA
SCHEMBL7360846 0.80 KDM4E (0.64) KDM4EALDH1A1TDP1MAPTGAA
SCHEMBL702118 0.78 TAS1R3 (0.57) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL38659004 0.78 TAS1R3 (0.57) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL7799940 0.78 KDM4E (0.50) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL6813093 0.77 HDAC1 (0.54) ALDH1A1SMN1; SMN2NPC1POLBLMNA
SCHEMBL8402587 0.77 LMNA (0.53) KDM4EALDH1A1TDP1ARMAPT
SCHEMBL11679419 0.77 AR (0.51) KDM4EALDH1A1TDP1ARMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096768-A ADMINISTERING A 3, 5, 6-SUBSTITUTED PHENYL COMPOUND FOR THE TREATMENT OF INFLAMMATION AND AUTOIMMUNE DISORDERS RHONE-POULENC RORER LIMITED (GB) 2000-08-01 US disclosed
US-5935978-A Compounds containing phenyl linked to aryl or heteroaryl by an aliphatic- or heteroatom-containing linking group RHONE-POULENC RORER LIMITED (GB) 1999-08-10 US disclosed
US-5840724-A COMPOUNDS FOR TUMOR NECROSIS FACTOR OR ENZYME INHIBITORS OF PHOSPHODIESTERASES RHONE-POULENC RORER LIMITED (GB) 1998-11-24 US disclosed
US-5698711-A INHIBITORS OF TUMOR NECROSIS FACTOR, CYCLIC ADENOSINE-3*,5*-MONOPHOSPHATE PHOSPHODIESTERASE AND EOSINOPHILS RHONE-POULENC RORER LIMITED (GB) 1997-12-16 US disclosed
US-5679696-A FOR INHIBITING TUMOR NECROSIS FACTOR; ENZYME INHIBITORS RHONE-POULENC RORER LIMITED (GB) 1997-10-21 US disclosed