SCHEMBL7432199

SCHEMBL7432199

O=C(O)c1ccc(N2CCOCC2)c(NC(=O)C(CS)Cc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.56
POLB P06746 1/20 0.52
TSHR P16473 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 3/20 0.47
KCNQ2 O43526 1/20 0.46
LMNA P02545 2/20 0.45
FOLH1 Q04609 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
KDM1A O60341 2/20 0.44
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
KDM1B Q8NB78 2/20 0.44
RCOR1 Q9UKL0 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440859 0.91 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP3A4KMT2AKCNQ2
SCHEMBL7433764 0.90 KMT2A (0.50) ALDH1A1POLBTSHRKMT2AKCNQ2
SCHEMBL7438709 0.78 MME (0.54) ALDH1A1KMT2AFOLH1HPGDMEN1
SCHEMBL7435482 0.78 KMT2A (0.56) ALDH1A1POLBTSHRNPSR1CYP1A2
SCHEMBL9456711 0.77 MEN1 (0.54) ALDH1A1KMT2AFOLH1HPGDGAA
SCHEMBL7434266 0.77 MME (0.57) ALDH1A1KMT2ALMNAFOLH1HPGD
SCHEMBL19084698 0.77 KDM1A (0.67) ALDH1A1POLBTSHRNPSR1CYP1A2
SCHEMBL7438991 0.77 MAPT (0.49) ALDH1A1CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL7432434 0.76 MAPT (0.48) ALDH1A1POLBCYP1A2CYP3A4CYP2C19
SCHEMBL7433690 0.75 MME (0.51) ALDH1A1KMT2AFOLH1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210266-A Analgesic enkephalinase inhibitors DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-05-11 US disclosed
US-5179125-A Analgesics DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1993-01-12 US disclosed
EP-0318859-A2 N-substituted mercaptopropanamide derivatives Dainippon Pharmaceutical Co., Ltd. (JP) 1989-06-07 EP disclosed