SCHEMBL7435909

SCHEMBL7435909

COc1cccc(OC)c1-c1nnn(CC(=O)C(CC(=O)O)NC(=O)OCc2ccccc2)n1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.51
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CASP1 P29466 16/20 0.48
TP53 P04637 1/20 0.46
ITGA4 P13612 1/20 0.44
ITGB7 P26010 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439044 0.90 CYP1A2 (0.46) CASP3CYP1A2CYP2C9CYP2C19CASP1
SCHEMBL7435530 0.88 CYP1A2 (0.63) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7431720 0.87 CASP1 (0.55) CASP3CYP1A2CYP2C9CYP2C19CASP1
SCHEMBL7429152 0.86 CYP1A2 (0.60) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7440449 0.85 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7677872 0.85 CASP1 (0.53) CASP3CASP1
SCHEMBL7434939 0.85 SMN1; SMN2 (0.57) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7439324 0.85 CYP1A2 (0.54) CYP1A2CYP2C9CYP2C19CASP1TP53
SCHEMBL7679972 0.84 CASP3 (0.48) CASP3CASP1
SCHEMBL7426313 0.84 CYP1A2 (0.53) CYP1A2CYP2C9CYP2C19CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US claimed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP claimed
US-5710153-A INTERLEUKIN CONVERTING ENZYME INHIBITORS ONO PHRAMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed
EP-0761680-A2 Tetrazole compounds having Interleukin-1beta converting enzyme inhibitory activity ONO PHARMACEUTICAL CO., LTD. (JP) 1997-03-12 EP disclosed