SCHEMBL7436632

SCHEMBL7436632

COc1ccc(-c2ccc(Cc3nc4c(ncn4C(C)CCCc4ccccc4)c(=O)[nH]3)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.53
ADORA3 P0DMS8 1/20 0.47
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
HPGD P15428 4/20 0.44
HSD17B10 Q99714 2/20 0.44
HTT P42858 2/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
BRS3 P32247 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 3/20 0.39
CCNB2 O95067 2/20 0.39
CDK1 P06493 2/20 0.39
CCNB1 P14635 2/20 0.39
CCNB3 Q8WWL7 2/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6051959 0.90 PDE2A (0.63) PDE2AADORA3KDM4ELMNAPOLB
SCHEMBL7502873 0.88 HPGD (0.44) PDE2AKDM4EALDH1A1HPGDHSD17B10
SCHEMBL7436563 0.87 PDE2A (0.57) PDE2AADORA3CCNB2CDK1CCNB1
SCHEMBL7442300 0.87 PDE2A (0.57) PDE2AADORA3KMT2ACCNE2CCNE1
SCHEMBL6051965 0.87 PDE2A (0.57) PDE2AADORA3HPGDMAPTPOLB
SCHEMBL6052132 0.86 PDE2A (0.51) PDE2AADORA3KDM4EALDH1A1HPGD
SCHEMBL6051979 0.86 PDE2A (0.53) PDE2AADORA3CCNB2CDK1CCNB1
SCHEMBL7440929 0.82 PDE2A (0.54) PDE2ACCNE2CCNE1CDK2
SCHEMBL7355722 0.81 ADORA3 (0.48) PDE2AADORA3KDM4EALDH1A1HPGD
SCHEMBL7442320 0.81 PDE2A (0.52) PDE2AADORA3KDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861396-A CARDIOVASCULAR DISORDERS AND UROGENITAL SYSTEMS BAYER AKTIENGESELLSCHAFT (DE) 1999-01-19 US disclosed
EP-0771799-A1 Purin-6-one derivatives BAYER AG (DE) 1997-05-07 EP disclosed