SCHEMBL7436833

SCHEMBL7436833

COc1ccc(-c2csc(C(N)=O)n2)c(Cl)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
SCN9A Q15858 1/20 0.40
MEN1 O00255 4/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
POLB P06746 2/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
THRB P10828 2/20 0.39
ATP4A P20648 2/20 0.39
ATP4B P51164 2/20 0.39
HSD17B10 Q99714 2/20 0.38
AMY1A P0DUB6 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435953 0.85 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
SCHEMBL7435945 0.80 ALDH1A1 (0.40) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
SCHEMBL6689068 0.78 CYP1A1 (0.64) ALDH1A1KDM4ESMN1; SMN2CYP3A4CYP2D6
SCHEMBL7430437 0.76 THRB (0.43) ALDH1A1CYP3A4CYP2D6CYP2C9SCN9A
SCHEMBL6687492 0.76 MEN1 (0.62) ALDH1A1KDM4ESMN1; SMN2CYP3A4CYP2D6
SCHEMBL7432599 0.74 HTR2C (0.60) ALDH1A1KDM4ESMN1; SMN2LMNACYP3A4
SCHEMBL2958088 0.73 KMT2A (0.47) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
Hydrochloric Acid SCHEMBL4501141 0.72 KMT2A (0.46) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
SCHEMBL3602404 0.72 KMT2A (0.45) ALDH1A1KDM4ESMN1; SMN2LMNAMEN1
SCHEMBL3580803 0.72 PDE4B (0.42) ALDH1A1KDM4ESMN1; SMN2LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506194-B1 4-aryl-thiazole or imidazole derivatives AKZO NOBEL NV (NL) 1996-08-21 EP disclosed
US-5462959-A 4-aryl-imidazole derivatives AKZO N.V. (NL) 1995-10-31 US disclosed
US-5254575-A 4-aryl-thiazole derivatives AKZO N.V. (NL) 1993-10-19 US disclosed
EP-0506194-A1 4-aryl-thiazole or imidazole derivatives Akzo Nobel N.V. (NL) 1992-09-30 EP disclosed