SCHEMBL7437151

SCHEMBL7437151

COc1ccccc1OCC(=O)NC(CC(C)C)C(=O)NC(Cc1ccccc1)C(=O)CSCc1ccco1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
PTPN1 P18031 2/20 0.43
CASP1 P29466 5/20 0.43
CASP3 P42574 5/20 0.43
CASP7 P55210 5/20 0.43
CASP8 Q14790 5/20 0.43
CASP6 P55212 3/20 0.43
PSMB5 P28074 2/20 0.43
PSMB1 P20618 1/20 0.42
PSMB2 P49721 1/20 0.42
TSHR P16473 1/20 0.42
REN P00797 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
FCER2 P06734 1/20 0.41
CAPN1 P07384 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437142 1.00 HPGD (0.46) HPGDPTPN1CASP1CASP3CASP7
SCHEMBL7341642 0.93 HPGD (0.53) HPGDTSHRKDM4EALDH1A1LMNA
SCHEMBL7341662 0.93 HPGD (0.53) HPGDTSHRKDM4EALDH1A1LMNA
SCHEMBL8683165 0.91 MEN1 (0.43) HPGDPTPN1CASP1CASP3CASP7
SCHEMBL8887573 0.91 MEN1 (0.43) HPGDPTPN1CASP1CASP3CASP7
SCHEMBL7303784 0.90 ALDH1A1 (0.49) HPGDPTPN1CASP1CASP3CASP7
SCHEMBL7303797 0.90 ALDH1A1 (0.49) HPGDPTPN1CASP1CASP3CASP7
SCHEMBL7436014 0.88 HPGD (0.46) HPGDCASP1CASP3CASP7CASP8
SCHEMBL7436020 0.88 HPGD (0.46) HPGDCASP1CASP3CASP7CASP8
SCHEMBL7437147 0.88 HPGD (0.45) HPGDPTPN1PSMB5PSMB1PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed