SCHEMBL7303784

SCHEMBL7303784

CC(C)C[C@H](NC(=O)COc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)CSCc1ccco1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
USP2 O75604 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
PTPN1 P18031 3/20 0.46
REN P00797 3/20 0.46
CASP3 P42574 5/20 0.45
PSMB5 P28074 2/20 0.45
PSMB1 P20618 1/20 0.45
PSMB2 P49721 1/20 0.45
CASP1 P29466 4/20 0.43
CASP7 P55210 4/20 0.43
CASP6 P55212 4/20 0.43
CASP8 Q14790 4/20 0.43
CTSD P07339 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303797 1.00 ALDH1A1 (0.49) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7435245 0.94 GPR34 (0.47) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7444214 0.94 ALDH1A1 (0.46) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7444208 0.94 ALDH1A1 (0.46) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7435258 0.94 GPR34 (0.47) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7301641 0.92 ALDH1A1 (0.48) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7301631 0.92 ALDH1A1 (0.48) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7350634 0.91 ALDH1A1 (0.58) ALDH1A1USP2POLBMAPTHPGD
SCHEMBL7437151 0.90 HPGD (0.46) ALDH1A1HPGDPTPN1RENCASP3
SCHEMBL7437142 0.90 HPGD (0.46) ALDH1A1HPGDPTPN1RENCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed