SCHEMBL7437423

SCHEMBL7437423

CC(C)(C)OC(=O)NC(C(=O)c1ccccc1)C(O)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 6/20 0.47
PPARG P37231 5/20 0.47
PPARD Q03181 2/20 0.47
TRPA1 O75762 2/20 0.44
GABRB1 P18505 1/20 0.44
GABRB2 P47870 1/20 0.44
CTSK P43235 3/20 0.43
CTSS P25774 3/20 0.43
ATM Q13315 1/20 0.43
ACE P12821 1/20 0.43
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
APP P05067 1/20 0.41
KLK5 Q9Y337 1/20 0.41
IDO1 P14902 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438625 0.87 TRPA1 (0.44) PPARAPPARGPPARDTRPA1GABRB1
SCHEMBL7438422 0.85 TRPA1 (0.57) PPARAPPARGPPARDTRPA1CTSK
SCHEMBL8283003 0.85 TRPA1 (0.57) PPARAPPARGPPARDTRPA1CTSK
SCHEMBL7441717 0.85 TSHR (0.43)
SCHEMBL29244798 0.84 PPARA (0.50) PPARAPPARGPPARDGABRB1GABRB2
SCHEMBL29244796 0.84 PPARA (0.50) PPARAPPARGPPARDGABRB1GABRB2
SCHEMBL7106002 0.80 CTSK (0.47) PPARAPPARGTRPA1CTSKCTSS
SCHEMBL7106006 0.80 CTSK (0.47) PPARAPPARGTRPA1CTSKCTSS
SCHEMBL23619006 0.79 PPARA (0.48) PPARAPPARGPPARDGABRB1GABRB2
SCHEMBL15432503 0.79 PPARA (0.48) PPARAPPARGPPARDGABRB1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed