SCHEMBL7437478

SCHEMBL7437478

COC(=O)N1Cc2ccccc2CCC1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 4/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 2/20 0.43
CHEK1 O14757 1/20 0.43
JAK2 O60674 1/20 0.43
ITGB3 P05106 1/20 0.42
ITGB1 P05556 1/20 0.42
ITGAV P06756 1/20 0.42
ITGA5 P08648 1/20 0.42
ITGA4 P13612 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MTNR1A P48039 2/20 0.40
MTNR1B P49286 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7435800 0.82 NR1D1 (0.51) ALDH1A1NPSR1KMT2AMEN1MTNR1A
SCHEMBL31759059 0.78 TSHR (0.39) ACEALDH1A1SMN1; SMN2ITGB3ITGB1
SCHEMBL10824345 0.77 ACE (0.79) ACE
SCHEMBL10824344 0.77 ACE (0.79) ACE
SCHEMBL16267600 0.74 ACE (0.43) ACEPOLBTDP1
SCHEMBL30801141 0.74 ACE (0.43) ACEPOLBTDP1
SCHEMBL9471352 0.74 ACE (0.45) ACE
SCHEMBL4627296 0.74 ACE (0.60) ACEALDH1A1POLBCHEK1JAK2
SCHEMBL5720519 0.74 ACE (0.60) ACEALDH1A1POLBCHEK1JAK2
SCHEMBL7274651 0.72 ACE (0.62) ACEPOLBNPSR1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670310-B1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants LILLY CO ELI (US) 1998-09-02 EP disclosed
US-5578574-A THROMBIN INHIBITORS OR ANTICOAGULANTS ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
EP-0672665-A1 Antithrombotic agents ELI LILLY AND COMPANY (US) 1995-09-20 EP disclosed
EP-0670310-A1 Bisulfite adducts of arginine aldehydes useful as thrombin inhibitors and as anticoagulants ELI LILLY AND COMPANY (US) 1995-09-06 EP disclosed