SCHEMBL7437828

SCHEMBL7437828

CC(C)Cn1c(=O)cc(C(=O)O)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.62
ALDH1A1 P00352 6/20 0.62
HSD17B10 Q99714 2/20 0.62
GAA P10253 2/20 0.62
HTR3E A5X5Y0 6/20 0.58
HTR3B O95264 6/20 0.58
HTR3A P46098 6/20 0.58
HTR3D Q70Z44 6/20 0.58
HTR3C Q8WXA8 6/20 0.58
HPGD P15428 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPT P10636 3/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HSP90AA1 P07900 1/20 0.45
ALOX15 P16050 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437043 0.86 HTR3E (0.61) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7436539 0.84 ALDH1A1 (0.67) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7434216 0.81 KDM4E (0.64) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7429056 0.79 ALDH1A1 (0.82) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7438285 0.79 ALDH1A1 (0.68) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7437593 0.78 ALDH1A1 (0.63) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7430518 0.78 HTR3E (0.56) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL7435320 0.77 ALDH1A1 (0.61) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL2921888 0.75 KDM4E (0.59) KDM4EALDH1A1HSD17B10GAAHTR3E
SCHEMBL2794759 0.75 KDM4E (0.56) KDM4EALDH1A1HSD17B10GAAHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed