SCHEMBL7435320

SCHEMBL7435320

CCCCCCn1c(=O)cc(C(=O)O)c2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
HTR3E A5X5Y0 4/20 0.61
HTR3B O95264 4/20 0.61
HTR3A P46098 4/20 0.61
HTR3D Q70Z44 4/20 0.61
HTR3C Q8WXA8 4/20 0.61
PSEN1 P49768 4/20 0.58
PSEN2 P49810 4/20 0.58
APH1B Q8WW43 4/20 0.58
NCSTN Q92542 4/20 0.58
APH1A Q96BI3 4/20 0.58
PSENEN Q9NZ42 4/20 0.58
KDM4E B2RXH2 4/20 0.58
GAA P10253 1/20 0.58
HSD17B10 Q99714 1/20 0.58
MAPT P10636 1/20 0.55
HTT P42858 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
CNR2 P34972 1/20 0.54
LMNA P02545 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7437593 0.99 ALDH1A1 (0.63) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7438285 0.95 ALDH1A1 (0.68) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7434216 0.89 KDM4E (0.64) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7436539 0.83 ALDH1A1 (0.67) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL9262842 0.82 ALDH1A1 (0.89) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL9254043 0.82 ALDH1A1 (0.89) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL30197876 0.82 ALDH1A1 (0.89) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7437043 0.80 HTR3E (0.61) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7435807 0.80 HTR3E (0.64) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7429517 0.79 KDM4E (0.55) ALDH1A1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed