SCHEMBL7437922

SCHEMBL7437922

CC(C)Cc1ccc(C(=O)CNC(=O)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KMT2A Q03164 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
MEN1 O00255 2/20 0.50
ALOX12 P18054 1/20 0.50
GPR139 Q6DWJ6 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
PPARG P37231 1/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
TAOK1 Q7L7X3 1/20 0.47
TAOK3 Q9H2K8 1/20 0.47
DPP4 P27487 1/20 0.47
LMNA P02545 3/20 0.47
MAPT P10636 2/20 0.47
SIGMAR1 Q99720 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557928 0.84 MEN1 (0.61) ALDH1A1KMT2ASMN1; SMN2MEN1CYP1A2
SCHEMBL23894858 0.83 HDAC1 (0.65) PPARGHDAC1HDAC6RAB9ALMNA
SCHEMBL3231208 0.82 ALDH1A1 (0.68) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL7432438 0.82 RAB9A (0.59) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL23014122 0.81 KMT2A (0.50) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL27855167 0.81 ESRRG (0.67) KMT2ASMN1; SMN2MEN1HDAC1HDAC6
Methane SCHEMBL11380092 0.81 ALDH1A1 (0.66) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL23014433 0.80 CES1 (0.59) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL28483353 0.80 ALDH1A1 (0.73) ALDH1A1KMT2ASMN1; SMN2MEN1ALOX12
SCHEMBL23014500 0.78 SIGMAR1 (0.56) KMT2AHDAC1HDAC6SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4453003-A ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS UMEZAWA HAMAO (JP) 1984-06-05 US disclosed
US-4391986-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediates therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-07-05 US disclosed
US-4281180-A Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1981-07-28 US disclosed