SCHEMBL7438523

SCHEMBL7438523

CCOC(=O)c1cnc2nc(CC)cc(N(C)c3ccc(-c4ccccc4-c4nnn[nH]4)cc3)n12

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.38
AGTR1 P30556 10/20 0.34
AGTR2 P50052 5/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440881 0.93 AGTR1 (0.36) AGTR1AGTR2
SCHEMBL7444851 0.91 AGTR1 (0.31) AGTR1AGTR2
SCHEMBL7442523 0.90 HSP90AA1 (0.32)
SCHEMBL7433640 0.85 AGTR1 (0.31) AGTR1AGTR2
SCHEMBL7427100 0.83 AGTR1 (0.32) AGTR1AGTR2
SCHEMBL7438663 0.83 KDM4E (0.43) AGTR1AGTR2
SCHEMBL7438511 0.82 AGTR1 (0.44) IDO1AGTR1AGTR2
SCHEMBL7429883 0.82
SCHEMBL7440495 0.81 TGFBR1 (0.36) AGTR1AGTR2
SCHEMBL7442759 0.79 AGTR1 (0.33) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed